KYLE, Donald J.,GOEHRING, R. Richard,FUNDYTUS, Marian E.
申请号:
AU2012251956
公开号:
AU2012251956A1
申请日:
2012.11.13
申请国别(地区):
AU
年份:
2012
代理人:
摘要:
#$%^&*AU2012251956A120121206.pdf#####ABSTRACT The present invention is directed to Buprenorphine Analog compounds of the 2 3 3a 3b Formula I, Formula II or Formula III shown below, wherein R1, R2 , R8, R3, Ra, R , X, Z and Y are as defined herein. N R 3 &RZ R2 H3CO O OCHa 5 (1) N "R R 3" &~~~R3b z0YR x O OCH3 (II) N R R3aa Z0 R2 R8 X0 OCHa (III) 10 Compounds of the Invention are useful for treating pain and other conditions modulated by activity of opioid and ORLI receptors. 1011995v1