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Inhibitors of Histone demethylase
专利权人:
CELGENE QUANTICEL RESEARCH; INC.
发明人:
申请号:
ARP170101007
公开号:
AR108286A1
申请日:
2017.04.19
申请国别(地区):
AR
年份:
2018
代理人:
摘要:
1. Claim 1: compound (1) with formula structure,Where R1 is halogen, ch83222; G, NHg or og, where G is hydrogen, tar, o-x-y, where x is hydrogen or tar-c8321;E replace aralquilo, replace aralquilo, replace aralquenilo, replace aralquinilo, replace aralquinilo, replace carbocyclo, replace heterosexual, replace heterosexual, replace heterosexual, Alternative allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic allylic 2-alternative dihydrofluoroalkanes,Alternative phenyl substitute, pyridine substitute, alternative tetrahydroquinol substitute, alternative tetramethylenedioxy substitute, alternative dioxin substitute, or alternative sulfur phosphorus substitute, - r74955-or74919;-R -OC (O) -R-R -OC (O) -OR-R -OC (O) -N (R)-R -N (R)-R -C (O) R-R -C (O) OR-R -O-R -C (O) N (R)-R -N (R) C (O) OR-R -N (R) C (O) R-R -N (R) S (O) R-R -S (O) OR-R -S (O) ORo -R -S (O) N (R)a. Each r74919 is independent of hydrogen, tar, fluoropropyl, CYCLOPROPYLENE, CYCLOPROPYLENE, arilo, aralquilo, isopropyl, isopropyl allyl, isopropylene or isopropenylene, and each r74955 is independent of a direct chain or a tar or a straight line or a separated daughter; Each r758080 is a tar or tonsil or branch chain; t is 1 or 2; R 2 is halogen or cf832323;R83099 is hydrogen, methyl, ethyl, isopropyl, t-butilo, chf832222;CH₂F, CF₃,CH OH CHCH OH o C (CH) OHReivindicación 1: Un compuesto que tiene la estructura de fórmula (1), donde R¹ es halógeno, CH₂G, NHG o OG, donde G es hidrógeno, alquilo, o -X-Y, en el cual X es hidrógeno o alquileno -C₁, e Y es aralquilo opcionalmente sustituido, aralquenilo opcionalmente sustituido, aralquinilo opcionalmente sustituido, carbociclilo opcionalmente sustituido, carbociclilalquilo opcionalmente sustituido, heteroc
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