您的位置: 首页 > 农业专利 > 详情页

DERIVADO DE AMINOPIRAZOL.
专利权人:
F. HOFFMAN-LA ROCHE AG
发明人:
HIROSATO EBIIKE,TADAKATSU HAYASE,LISHA WANG,NAOKI TAKA,MASAYUKI OHMORI,KYOKO TAKAMI,MASAYUKI MATSUSHITA,IKUMI HYODO,MASAMI KOCHI,HIROKI NISHII,YOSHITO NAKANISHI,TOSHIYUKI MIO,WEILI ZHAO
申请号:
MX2012001653
公开号:
MX2012001653A
申请日:
2010.08.05
申请国别(地区):
MX
年份:
2012
代理人:
摘要:
A compound represented by formula (I) or a pharmacologically acceptable salt thereof, which can inhibit a fibroblast growth factor receptor (FGFR) family kinase in cancer tissues. (In the formula, A represents a 5- to 10-membered heteroaryl group, or a C6-10 aryl group; R1 and R2 independently represent H, OH, X, CN, NO2, a C1-4 haloalkyl group, a C1-6 alkyl group, or the like <;R1 and R2 together form a (substituted) 3- to 10-membered heterocyclyl group or a (substituted) 5- to 10-membered heteroaryl group>;; R3 represents H, a C1-5 alkyl group, a C6-10 aryl group, a C1-5 alkyl group, or a C1-4 haloalkyl group; and R4 represents H, X, a C1-3 alkyl group, a C1-4 haloalkyl group, OH, CN, NO2, or the like.).Se describen métodos para tratar cáncer al administrar un compuesto de la fórmula (I), (fórmula I) o una sal farmacéuticamente aceptable o solvato del mismo, en combinación con otros tratamientos de cáncer, en donde R1 es halo; R2 es halo; y Q es CH o N.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充