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FORMES CRISTALLINE ET AUTRES DE SELS D'ACIDE LACTIQUE 4-AMINO-5-FLUORO-3-[6-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]-1H-QUINOLIN-2-ONE
专利权人:
NOVARTIS AG
发明人:
OKHAMAFE, AUGUSTUS,CHOU, JOYCE,GULLAPALLI, RAMPURNA,HARWOOD, ERIC,RYCKMAN, DAVID,ZHU, SHUGUANG,SHANG, XIAO
申请号:
CA2609353
公开号:
CA2609353C
申请日:
2006.05.23
申请国别(地区):
CA
年份:
2015
代理人:
摘要:
The present invention relates to non-hydrate crystalline forms of 4-amino- 5-fluoro-3 -[6-(4-methylpiperazin- 1 -yl)- 1 H-benzimidazol-2-yl] - 1 H-quinolin-2-one lactic acid salts, solid pharmaceutical formulations containing the sameand methods of use. The present invention also relates to crystalline hydratesof 4-arnino-5-fiuoro-3-[6-(4- methylpiperazin-l-yl)-lH-benzimidazol-2-yl]-lH-quinolin-2-one lactic acid salts, pharmaceutical formulations containing thesame and methods of use related thereto. The present invention further relatesto crystalline solvates of 4-amino-5-fluoro-3-[6-(4- methylpiperazin-l-yl)-lH-benzimidazol-2-yl]-lH-quinolin-2-one lactic acid salts.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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