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COMPOUNDS WHICH HAVE ACTIVITY AT M₁ RECEPTOR AND THEIR USES IN MEDICINE
专利权人:
GLAXO GROUP LIMITED
发明人:
BUDZIK, BRIAN,COOPER, DAVID, GWYN,FORBES, IAN THOMSON,GARZYA, VINCENZO,JIN, JIAN,SHI, DONGCHUAN,SMITH, PAUL, WILLIAM,WALKER, GRAHAM
申请号:
MYPI 20080901
公开号:
MY148504A
申请日:
2006.09.27
申请国别(地区):
MY
年份:
2013
代理人:
摘要:
COMPOUNDS OF FORMULA (I) AND SALTS AND SOLVATES ARE PROVIDED: WHEREIN R⁴ IS FLUORO, R⁵ IS SELECTED FROM HYDROGEN, HALOGEN, CYANO, C₁-₆ALKYL, C₁-₆ALKYL SUBSTITUTED WITH ONE OR MORE FLUORINE ATOMS, C₁-₆ALKOXY, AND C₁-₆ALKOXY SUBSTITUTED WITH ONE OR MORE FLUORINE ATOMS, AND R⁶ IS SELECTED FROM HALOGEN, CYANO, C₁-₆ALKYL, C₁-₆ALKYL SUBSTITUTED WITH ONE OR MORE FLUORINE ATOMS, C₃ -₆CYCLOALKYL, C₃ -₆CYCLOALKYL SUBSTITUTED WITH ONE OR MORE FLUORINE ATOMS, C₁-₆ALKOXY AND C₁-₆ALKOXY SUBSTITUTED WITH ONE OR MORE FLUORINE ATOMS, AND Q IS HYDROGEN OR C₁-₆ALKYL. THE COMPOUNDS ARE EXPECTED TO BE USEFUL FOR THERAPY, FOR EXAMPLE IN THE TREATMENT OF PSYCHOTIC DISORDERS AND COGNITIVE IMPAIRMENT.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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