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"2- [4- (PYRAZOL-4-ILALKYL) PIPERAZIN-1-IL] -3-PHENYL PIRAZINS AND PYRIDINS AND 3- [4- (PIRAZOL-4-ILALKYL) PIPERAZIN-1-IL] -2-PHENYL PYRIDINS AS 5-HT7 "RECEPTOR ANTAGONISTS
专利权人:
ELI LILLY AND COMPANY
发明人:
VALENTINA O. BADESCU,ANNE MARIE CAMP,BARRY PETER CLARK,MICHAEL PHILIP COHEN,SANDRA ANN FILLA,PETER THADDEUS GALLAGHER,SARAH LYNNE HELLMAN,MICHAEL PHILIP MAZANETZ,MARTA MARIA PINEIRO-NUNEZ,JOHN MEHNERT
申请号:
BRPI0811446
公开号:
BRPI0811446A2
申请日:
2008.05.07
申请国别(地区):
BR
年份:
2014
代理人:
摘要:
The present invention provides selective 5-HT7 receptor antagonist compounds of Formula I and their use in the treatment of migraine, persistent pain, and anxiety: where A and B are each independently —C(H)═ or —N═, provided that at least one of A and B is —N═, n is 1-3, m is 0-3, and R1-4 are as defined herein.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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