2-[4-(PIRAZOL-4-ILOALKILO)PIPERAZYN-1-YLO]-3-FENYLO PIRAZYNY I PIRYDYNY I 3-[4-(PIRAZOL-4-ILOALKILO)PIPERAZYN-1-YLO]-2-FENYLO PIRYDYNY JAKO ANTAGONIŚĆI RECEPTORA 5-HT<;sub>;7<;/sub>;
BADESCU, VALENTINA O.,CAMP, ANNE MARIE,CLARK, BARRY PETER,COHEN, MICHAEL PHILIP,FILLA, SANDRA ANN,GALLAGHER, PETER THADDEUS,HELLMAN, SARAH LYNNE,MAZANETZ, MICHAEL PHILIP,PINEIRO-NUNEZ, MARTA MARIA,SCH
申请号:
PL08747748
公开号:
PL2155717T3
申请日:
2008.05.07
申请国别(地区):
PL
年份:
2013
代理人:
摘要:
The present invention provides selective 5-HT7 receptor antagonist compounds of Formula I and their use in the treatment of migraine, persistent pain, and anxiety: where A and B are each independently &mdash;C(H)&boxH; or &mdash;N&boxH;, provided that at least one of A and B is &mdash;N&boxH;, n is 1-3, m is 0-3, and R1-4 are as defined herein.