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SALES DE HIDROCLORURO DE 8-[{1-(3,5-BIS-(TRIFLUOROMETIL)FENIL)-ETOXI}-METIL]-8-FENIL-1,7-DIAZASPIRO[4.5]DECAN-2-ONA
专利权人:
OPKO HEALTH; INC.
发明人:
SHIH, NENG-YANG,PALIWAL, SUNIL,GUENTER, FRANK,MERGELSBERG, INGRID,HU, MENGWEI
申请号:
PE0007582014
公开号:
PE23292014A1
申请日:
2007.04.04
申请国别(地区):
PE
年份:
2015
代理人:
摘要:
(i) refers to a form of anhydrous Crystalline hydrochloride Salt of (5S, 8S) - 8 - [(1R) - 1 - (3,5-bis - (trifluoromethyl) phenyl) - ethoxy) - methyl] - 4 - phenyl - 1.7 - diazaspiro [4.5] - 2 - (Deccan Ona formula (i) which Presents a pattern of x-ray Powder diffraction Peaks that are present in the angles of difraccio N 2 Theta: 12.9 (S), (S), 15.4 20.2 17.3 (S), (S).Is also referred to the Crystalline forms (ii), (iii) and (iv) tosylate salt (5S, 8S) - 8 - [(1R) - 1 - (3,5-bis - (trifluoromethyl) phenyl) - ethoxy) - methyl] - 4 - phenyl - 1.7 - diazaspiro [4.5] decan 2 - onaREFERIDA A UNA FORMA (I) CRISTALINA ANHIDRA DE LA SAL DE HIDROCLORURO DE (5S,8S)-8-[{(1R)-1-(3,5-BIS-(TRIFLUOROMETIL)FENIL)-ETOXI}-METIL]-8-FENIL-1,7-DIAZASPIRO[4.5]DECAN-2-ONA (FORMULA I) QUE PRESENTA UN PATRON DE DIFRACCION DE POLVO DE RAYOS X QUE TIENE PICOS PRESENTES EN LOS ANGULOS DE DIFRACCION EN 2 THETA DE: 12,9 (S), 15,4 (S), 17,3 (S), 20,2 (S). TAMBIEN ESTA REFERIDA LAS FORMAS CRISTALINAS (II), (III) Y (IV) DE LA SAL TOSILATO DE (5S,8S)-8-[{(1R)-1-(3,5-BIS-(TRIFLUOROMETIL)FENIL)-ETOXI}-METIL]-8-FENIL-1,7-DIAZASPIRO[4.5]DECAN-2-ONA
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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