5,6-dihydro-4 - [(difluoroethyl) phenyl] -4h-pyrrolo [1,2-a] [1,4] benzodiazepine and 4- (difluoroethyl) phenyl-6h-pyrrolo [1] antifungal agents , 2-a] [1,4] benzodiazepine

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专利权人:

JANSSEN PHARMACEUTICA NV

发明人:

KELLY DE WIT,LIEVEN MEERPOEL,LOUIS JULES ROGER MARIE MAES

申请号：

BR112012030895

公开号：

BR112012030895A2

申请日:

2011.06.01

申请国别(地区):

BR

年份:

2016

代理人:

摘要：

The present invention concerns novel compounds of Formula (I): wherein R1, R2, R3, R4, R5 and R6 have the meaning defined in the claims. The compounds according to the present invention are active mainly against dermatophytes and systemic fungal infections. The invention further relates to processes for preparing such novel compounds, pharmaceutical compositions comprising said compounds as an active ingredient as well as the use of said compounds as a medicament.

来源网站：

中国工程科技知识中心

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http://www.ckcest.cn/home/