Antifungal 5,6-dihydro-4-[(difluoroethyl)phenyl]-4H-pyrrolo[1,2-α][1,4]benzodiazepine and 4-(difluoroethyl)phenyl-6H-pyrrolo[1,2-α][1,4]benzodiazepine derivatives
Lieven Meerpoel;Louis Jules Roger Marie Maes;Kelly de Wit
发明人:
Lieven Meerpoel,Louis Jules Roger Marie Maes,Kelly de Wit
申请号：
US13702361
公开号：
US09637490B2
申请日:
2011.06.01
申请国别(地区):
US
年份:
2017
代理人:
摘要：
The present invention concerns novel compounds of Formula (I):wherein R1, R2, R3, R4, R5 and R6 have the meaning defined in the claims. The compounds according to the present invention are active mainly against dermatophytes and systemic fungal infections. The invention further relates to processes for preparing such novel compounds, pharmaceutical compositions comprising said compounds as an active ingredient as well as the use of said compounds as a medicament.
