SUBSTITUTED TETRAHYDROPYRAN SPIRO PYRROLIDINONE AND PIPERIDINONE, PREPARATION AND THERAPEUTIC USE THEREOF

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专利权人:

SANOFI

发明人:

GAO, ZHONGLI,HARTUNG, RYAN,STEFANY, DAVID

申请号：

MYPI 2011002068

公开号：

MY150789A

申请日:

2009.12.04

申请国别(地区):

MY

年份:

2014

代理人:

摘要：

THE PRESENT DISCLOSURE RELATES TO A SERIES OF SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES OF FORMULA (I): WHEREIN R1, R2, M, N AND P ARE AS DESCRIBED HEREIN. MORE SPECIFICALLY, THE COMPOUNDS OF THIS INVENTION ARE MODULATORS OF H3 RECEPTORS AND ARE, THEREFORE, USEFUL AS PHARMACEUTICAL AGENTS, ESPECIALLY IN THE TREATMENT AND/OR PREVENTION OF A VARIETY OF DISEASES MODULATED BY H3 RECEPTORS INCLUDING DISEASES ASSOCIATED WITH THE CENTRAL NERVOUS SYSTEM. ADDITIONALLY, METHODS OF PREPARATION OF SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND INTERMEDIATES THEREFORE ARE DISCLOSED.

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