MEUTERMANS, WIM,SCHAFER, KARL,WEST, MICHAEL LEO,MULDOON, CRAIG,FOLEY, FIONA,BOULOC, NATALIE,TOMETZKI, GERALD
申请号：
ES12161249
公开号：
ES2445922T3
申请日:
2003.09.05
申请国别(地区):
ES
年份:
2014
代理人:
摘要：
A compound of the formula I which is a derivative of a furanosa form of a general formula I monosaccharide, ** Formula ** in which: n is 1, X is selected from: ** Formula ** R3 is selected from the group consisting of: C1 to C7 alkyl, C1 to C7 alkenyl, C1 to C7 alkynyl, C1a C7 heteroalkyl, C6 to C14 aryl, C3 to C14 heteroaryl, C6 to C14 arylalkyl, and C3 to C14 heteroarylalkyl, R4 is selected from the compound group by: C1 to C7 alkyl, C1 to C7 alkenyl, C1 to C7 alkynyl, C1a C7 heteroalkyl, C6 to C14 aryl, C3 to C14 heteroaryl, C6 to C14 arylalkyl, and C3 to C14 heteroarylalkyl, R5 is selected from the group consisting of: C1 to C7 alkyl, C1 to C7 alkenyl, C1 to C7 alkynyl, C1a C7 heteroalkyl, C6 to C14 aryl, C3 to C14 heteroaryl, C6 to C14 aryl alkyl or C3 to C14 heteroarylalkyl, C1 to C7 acyl, C6 to C14 arylacyl and C3 heteroarylacyl at C14, R2 is selected from - (C>； = O) -R3, - (C>； = O) -OR4, - (C>； = O) -NH.Un compuesto de la fórmula I que es un derivado de una forma de furanosa de un monosacárido defórmula general I,**Fórmula** en la que: n es 1, X se selecciona entre:**Fórmula** R3 se selecciona entre el grupo compuesto por: alquilo C1 a C7, alquenilo C1 a C7, alquinilo C1 a C7, heteroalquilo C1a C7, arilo C6 a C14, heteroarilo C3 a C14, arilalquilo C6 a C14 y heteroarilalquilo C3 a C14, R4 se selecciona entre el grupo compuesto por: alquilo C1 a C7, alquenilo C1 a C7, alquinilo C1 a C7, heteroalquilo C1a C7, arilo C6 a C14, heteroarilo C3 a C14, arilalquilo C6 a C14 y heteroarilalquilo C3 a C14, R5 se selecciona entre el grupo compuesto por: alquilo C1 a C7, alquenilo C1 a C7, alquinilo C1 a C7, heteroalquilo C1a C7, arilo C6 a C14, heteroarilo C3 a C14, arilalquilo C6 a C14 o heteroarilalquilo C3 a C14, acilo C1 a C7, arilacilo C6 aC14 y heteroarilacilo C3 a C14, R2 se selecciona entre -(C>；=O)-R3, -(C>；=O)-OR4, -(C>；=O)-NH.
