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Pyrazolidan compounds and their applications
专利权人:
INC.;ADURO BIOTECH
发明人:
ISMAILI, HOSSEIN,GILLARD, LAURA,ZAKY, MARIAM,RYBAK, TARAS,RAMTOHUL, YEEEMAN K.,LY, VU LINH,RAEPPEL, FRANCK,CIBLAT, STEPHANE,SUNG, LEONARD,ROBERTS, TUCKER CURRAN,KATIBAH, GEORGE EDWIN,NDUBAKU, CHUDIOBI
申请号:
ARP180102630
公开号:
AR113114A1
申请日:
2018.09.14
申请国别(地区):
AR
年份:
2020
代理人:
摘要:
1. Claim 1: a formula compound (1),1. A pharmaceutically acceptable salt, a pharmaceutically acceptable solution or a pharmaceutically acceptable hydrate, where y is - Cr n =;R1 is q1-t1 - (x1) 8345;;Q1 is link c832131 or lessor;a. Among them, c8321c8331832323 asphalt group is replaced by one or more independent halogenated group c18321c8331832626 asphalt substitutes;Alquenilo C83228331-832626;1. C 83228331 asphalt;Cyanogen, halide c8321c831832626,-Or695;Y-Nr.695;-R 739;;2T1 is cycloquilo c2238331;Arilo C832628331-8321;8320;3 to 12 members of isoprene, 5 to 10 members of isoprene, (= O) tar c833208331832323238331;-C (= O) - asphalt c8332083331;-C (= O) - 3-12 members heterosexual - C (= O) - 5-10 members heterosexual - nr7491931; r749595;-S(=O)8322;R74919-,-No. 7491; (= O) r74919 -,-No. 7491; (= O) No. 7491; - No. 7495;-No. 7491; (= O) No. 7491;-7491; (= O) 8322; - r7491;-C(=O)N7491;(=O)8322;-R7491;-No. 7491; (= O) 8322; - No. 7491;; No. r74955;-C(=O)N7491;R7495;o-S(=O)83222;n7491;R7495;Each X1 is selected independently from the group consisting of halide, cyanide, oxo, tar c8320331-c (= O) r758080;Lessor c832031c8331 ° - or758080;1.C83208C83331-83323C(=O)Or758080;1.C83208C83331-833230OC(=O)R758080;1. Lessor c832083315238nr7580; r74966;1. Lessor c8332083313523231n 83144r758080; r7496; r7496 ';1.C83208331C83323S(=O)8344R758080;1.C(=O)R758080;1.C(=O)NR7580;;R74966;1.C83208331°833230OC(=O)NR758080;R74966;1.C(=O)Or758080;Lessor c83320833135233808; (= O) 8322;; r758080;1.C8320833135238C(=O)NR758080;(=O)83222;;R758080;1. Loaner c83320833135233808; (= O) 8322;; n7580;; r749696; 1. Asphalt-c8320316c833231c (= O) n7580808; r74966;Lessor c833208331352323s (= O) 8322; = No. 7580808; r74966;Lessor c833208331c83331c238c (= nr758080); r74966;1.C(=NR 758080)NR 758080;And RS1,RS1 is apartment c833218331832626,Alquenilo C83228331-832626;1. C 83228331 asphalt;1.C83208331-83331-cycloquilo C832331-8328;1. Lessor c833208331c8331-arilo c833226833183218320;a. C833208331832316c-3 to 12 m
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