БЕЙКЕР Стефен Дж. (US),АКАМА Цутому (US),БЕЛЛИНГЕР-КАВАХАРА Кэролин (US),ЭРНАНДЕС Винсент С. (US),ХОУЛД Карин М. (US),ЛАЙДЕН Джеймс Дж. (US),МЕЙПЛЗ Керк Р. (US),ПЛАТТНЕР Джейкоб Дж. (US),САНДЕРЗ Вирдж
申请号：
RU2010133524/04
公开号：
RU2010133524A
申请日:
2010.08.10
申请国别(地区):
RU
年份:
2012
代理人:
摘要：
1. A compound having the following structure of formula (IIb):! ! where! R1b is selected from a negative charge, H and a salt counterion； ! R7b is selected from H, methyl, ethyl, and phenyl； ! R10b is selected from H, OH, NH2, SH, halogen, substituted or unsubstituted phenoxy, substituted or unsubstituted phenylalkyloxy, substituted or unsubstituted phenylthio, and substituted or unsubstituted phenylalkylthio； and! R11b is selected from H, OH, NH2, SH, methyl, substituted or unsubstituted phenoxy, substituted or unsubstituted phenylalkyloxy, substituted or unsubstituted phenylthio, and substituted or unsubstituted phenylalkylthio； ! provided that the compound is not a compound selected from the following compounds:! ； ； ； ； ； ； ； ； ； and. ! 2. The compound according to claim 1, where! R7b is selected from H； ! R10b is selected from substituted phenoxy, substituted or unsubstituted phenylalkyloxy, substituted or unsubstituted phenylthio, and substituted or unsubstituted phenylalkylthio； and! R11b is selected from H.! 3. The compound according to claim 1, where! R7b is selected from H； ! R10b is selected from phenoxy； and! R11b is selected from H.! 4. The compound according to claim 1, which is 5- (4-cyanophenoxy) -1,3-dihydro-1-hydroxy-2,1-benzoxaborol. ! 5. The compound according to claim 1, which is 5- (3,4-dicyanophenoxy) -1,3-dihydro-1-hydroxy-2,1-benzoxaborol. ! 6. A pharmaceutical preparation containing! a) a compound having a structure according to Formula (IIb):! ! where! R7b is selected from H, methyl, ethyl, and phenyl； ! R10b is selected from H, OH, NH2, SH, halogen, substituted or unsubstituted phenoxy, substituted or unsubstituted phenylalkyloxy, substituted or unsubstituted phenylthio, and substituted or unsubstituted phenylalkylthio； and! R11b is selected from H, OH, NH2, SH, methyl, substituted or unsubstituted phenoxy, substituted1. Соединение, имеющее следующую структуру формулы (IIb): ! ! где ! R1b выбран из отрицательного заряда, Н и солевог
