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2, 6-DIAMINO-PYRIMIDIN-5-YL-CARBOXAMIDES AS SYK OR JAK KINASES INHIBITORS
专利权人:
PORTOLA PHARMACEUTICALS; INC.
发明人:
BAUER, SHAWN M.,J. JIA, ZHAOZHONG,SONG, YONGHONG,XU, QING,MEHROTRA, MUKUND,ROSE, JACK W.,HUANG, WOLIN,VENKATARAMANI, CHANDRASEKAR,PANDEY, ANJALI
申请号:
MYPI 2010004846
公开号:
MY155639A
申请日:
2009.04.16
申请国别(地区):
MY
年份:
2015
代理人:
摘要:
THE PRESENT INVENTION IS DIRECTED TO COMPOUNDS OF FORMULA I-II AND PHARMACEUTICALLY ACCEPTABLE TAUTOMERS, SALTS, OR STEREOISOMERS THEREOF WHICH ARE INHIBITORS OF SYK AND/OR JAK KINASE. THE PRESENT INVENTION IS ALSO DIRECTED TO INTERMEDIATES USED IN MAKING SUCH COMPOUNDS, THE PREPARATION OF SUCH A COMPOUND, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH A COMPOUND, METHODS OF INHIBITION SYK AND/OR JAK KINASE ACTIVITY, METHODS OF INHIBITION THE PLATELET AGGREGATION, AND METHODS TO PREVENT OR TREAT A NUMBER OF CONDITIONS MEDIATED AT LEAST IN PART BY SYK AND/OR JAK KINASE ACTIVITY, SUCH AS CARDIOVASCULAR DISEASE, INFLAMMATORY DISEASE, AUTOIMMUNE DISEASE AND CELL PROLIFERATIVE DISORDER, THROMBOSIS, ALLERGY, ASTHMA, RHEUMATOID ARTHRITIS, LEUKEMIA, OR NON-HODGKIN’S LYMPHOMA. (NO SUITABLE FIGURE)
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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