DERIVATIVES OF BENZOTHIAZINES,PREPARATION THEREOF AND APPLICATION THEREOF AS DRUGS

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专利权人:

发明人:

PEREZ MICHEL,LAMOTHE MARIE,JUNQUERO DIDIER,RIVAL YVES

申请号：

IN7244/DELNP/2011

公开号：

IN2011DN07244A

申请日:

2011.09.21

申请国别(地区):

IN

年份:

2013

代理人:

摘要：

The object of the present invention is benzothiazine derivatives having the capability of inhibiting 11ß-HSD1 not only at an enzymatic level but also at a cell level. The compounds of the present invention are of general formula (I). Wherein notably R1 represents a hydrogen or OR1 represents an ester or an ether. R2 represents a naphthyl or a 1, 2, 3, 4-tetrahydro-naphthalene or a biphenyl or phenyl pyridine or a substituted phenyl. R3 represents a methyl or ethyl R4 and R4 represent a hydrogen.

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