DERIVATIVES OF BENZOTHIAZINES, PREPARATION THEREOF AND APPLICATION THEREOF AS DRUGS

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专利权人:

PIERRE FABRE MEDICAMENT

发明人:

PEREZ, MICHEL,LAMOTHE, MARIE,JUNQUERO, DIDIER,RIVAL, YVES

申请号：

MYPI 2011004096

公开号：

MY160819A

申请日:

2010.03.02

申请国别(地区):

MY

年份:

2017

代理人:

摘要：

THE OBJECT OF THE PRESENT INVENTION IS BENZOTHIAZINE DERIVATIVES HAVING THE CAPABILITY OF INHIBITING 11β-HSD1 NOT ONLY AT AN ENZYMATIC LEVEL BUT ALSO AT A CELL LEVEL.THE COMPOUNDS OF THE PRESENT INVENTION ARE OF GENERAL FORMULA (I): WHEREIN NOTABLY R1 REPRESENTS A HYDROGEN OR OR1 REPRESENTS AN ESTER OR AN ETHER. R2 REPRESENTS A NAPHTHYL OR A 1,2,3,4-TETRAHYDRO- NAPHTHALENE OR A BIPHENYL OR PHENYL PYRIDINE OR A SUBSTITUTED PHENYL R3 REPRESENTS A METHYL OR ETHYL R4 AND R’4 REPRESENT A HYDROGEN.

来源网站：

中国工程科技知识中心

来源网址：

http://www.ckcest.cn/home/