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Quinase thyroid inhibitor similar to FMS
专利权人:
3SM BIOTRON INC.
发明人:
HSU, JIUNN YUAN,CHEN, I,CHUN - LY, TAI WEI,CHEN, TSUNG,CHIH - CHEN, JUNG-HSIANG
申请号:
ARP180100838
公开号:
AR111401A1
申请日:
2018.04.04
申请国别(地区):
AR
年份:
2019
代理人:
摘要:
1. Requirement 1: Compounds conforming to (1) formula.(2)(3) or (4)Where Y is [P].8345;,Where P is-N-O-OX is [Q] 8345;Q is -C832222-,- No.- It's...- Yes.- SO832222-O-N-asphalt; N is 0 or 1; R1 represents monkeys-Say...3-or 4-substitutes and chooses from halogens.- No. 8322;- CN, copilo, alquenilo, halogalo, NHR74919,N (R74955) 832222;- Or7491,3, 4, 5 or 6 members of cyclopentadienol, 3, 4, 5, 6, non-cyclopentadienol, which contains one or two hetero-atoms selected from N, O and S, Arilo or heterogeneity; R74919 is H, tar, ene, halogen, hydroxyl-OH, -NO832222 or phenyl; R749595 tar, ene or halogen; R2 ES-NR7496; -R74977;- 0 - tar, C (= O) - 5 or 6 O - C (= O) - heterosexual, 5 or 6 members; R749669 is OH, tar, alkali, Arilo, heterosexual, heterosexual, R7491; R749779;- Asphalt-N (R74955) 8322;- Rental - Or 7580,- Heterosexuals renting 5 to 6 members, heterosexuals of 5 to 6 members, heterosexuals of 5 to 6 members, heterosexuals of 5 to 6 members, or heterosexuals with at least one N; R74977 is H, coagulant, Alquenilo or Arilo; R749696; R74977 forms 3 to 8 members of heterosexuals or heterosexuals with N, optionally. E. Solid or C83218331832323 alkyl group, C832183318323AOC, R758080 H, tar, halogen, halogen, or phenyl; R3 H, tar, Alquenilo, halogen, or CN, N8322O NOC832222;1. When tar or Alquenilo is not replaced or replaced by halogen, hydroxyl, amino or nitrogen, nor is it replaced or replaced by halogen with cyclopropyl or isocyclopropyl;- No. 8322;- CN, copilo, alquenilo. -NHR 749191,N (R74955) 8322O-Or74919;If P-CH and N are 1, R1 is not CL, or solution, stain, disinfection, corresponding substance, or salt with acceptable efficacy.Reivindicación 1: Un compuesto que responde a la fórmula (1), (2), (3) ó (4), donde Y es [P]ₙ, donde P es -CH-, -N- o -O-; X es [Q]ₙ, donde Q es -CH₂-, -N-, -O-, -S-, -SO₂- o -N-alquilo; n es 0 ó 1; R¹ representa mono-, di-, tri- o tetra-sustitución y se selecciona entre halógeno, -OH, -NH₂, -NO₂, -CN, alquilo, alquenilo, haloalquilo,
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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