DERIVES DE XANTHINE ET LEURS UTILISATIONS EN TANT QU'INHIBITEURS DE BROMODOMAINES DE PROTEINES BET

• 收藏
• 分享

专利权人:

UNIVERSITE D'AIX NARSEILLE;INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM);CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE

发明人:

BETZI, STEPHANE,COMBES, SEBASTIEN,COLLETTE, YVES,HOFFER, LAURENT,MORELLI, XAVIER,RAUX, BRIGIT,ROCHE, PHILIPPE,VOITOVICH, IULIIA

申请号：

CA3081753

公开号：

CA3081753A1

申请日:

2018.11.06

申请国别(地区):

CA

年份:

2019

代理人:

摘要：

The present invention relates to a compound having the following formula (I): (I) wherein: - R is a (C1-C6)alkyl group；- R'' is preferably H；- Ar is a (C5-C12)arylene radical；- X1 is -C(=O)- or -SO2-； and- R' is chosen from the group consisting of possibly substituted (C1-C6)alkyl, heteroaryl, (C5-C12)aryl, and (hetero)cycloalkyl groups, or a pharmaceutically acceptable salt and/or tautomeric form thereof, or its racemates, diastereomers or enantiomers.

来源网站：

中国工程科技知识中心

来源网址：

http://www.ckcest.cn/home/