5-biphenyl-4-heteroarylcarbonylamino-pentanoic acid derivatives as neprilysin inhibitors
- 专利权人:
- LLC;Theravance Biopharma R&D IP
- 发明人:
- Fleury, Melissa,Beausoliel, Anne-Marie,Hughes, Adam D.,Long, Daniel D.,Wilton, Donna A.A.
- 申请号:
- AU2015211041
- 公开号:
- AU2015211041B2
- 申请日:
- 2015.01.29
- 申请国别(地区):
- AU
- 年份:
- 2018
- 代理人:
- 摘要:
- In one aspect, the invention relates to compounds having the formula (I): where R
- 来源网站:
- 中国工程科技知识中心
相关发明人
相关专利
- 5-BIPHENYL-4-HETEROARYLCARBONYLAMINO-PENTANOIC ACID DERIVATIVES AS NEPRILYSIN INHIBITORS
- 5-BIPHENYL-4-HETEROARYLCARBONYLAMINO-PENTANOIC ACID DERIVATIVES AS NEPRILYSIN INHIBITORS
- 5-BIPHENYL-4-HETEROARYLCARBONYLAMINO-PENTANOIC ACID DERIVATIVES AS NEPRILYSIN INHIBITORS
- CRYSTALLINE (2S,4R)-5-(5'-CHLORO-2'-FLUORO-[1,1'-BIPHENYL]-4-YL)-2-(ETHOXYMETHYL)-4-(3-HYDROXYISOXAZOLE-5-CARBOXAMIDO)-2-METHYLPENTANOIC ACID AND USES THEREOF
- (2S, 4R)-5-(5-CHLORO-2-FLUOROBIPHENYL-4-YL)-2-ETHOXYOXALYLAMINO)-2-HYDROXYMETHYL-2-METHYLPENTANOIC ACID AS NEPRILYSIN INHIBITOR


