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compounds and pharmaceutical composition
专利权人:
PHENEX PHARMACEUTICALS AG
发明人:
Christian Gege,Christoph Steeneck,Gerald Kleyman,Olaf Kinzel,Thomas Hoffmann
申请号:
BR112014029868
公开号:
BR112014029868A2
申请日:
2013.05.29
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
1/1 Summary "Compounds and Pharmaceutical Composition" The invention provides modulators for the nuclear receptor orphan rorum and methods for the treatment of rhetorically mediated diseases by the administration It is these new modulators of rorý³ to a human being or a mammal who needs it. Specifically, the present invention provides a carboxamide or sulfonamide containing cyclic compounds of formula (1), (1 '), (100), (100'), (200) and (200 '),,, and the enantiomers, diastereoisomers, tautomers, n-oxides, solvates and pharmaceutically acceptable salts thereof.1 / 1 resumo “compostos, e, composiã‡ãƒo farmacãšuticaâ€� a invenã§ã£o fornece moduladores para o receptor nuclear ã³rfã£o rorî³ e mã©todos para o tratamento de doenã§as mediadas por rorî³ pela administraã§ã£o desses novos moduladores do rorî³ a um ser humano ou um mamã­fero que necessita disso. especificamente, a presente invenã§ã£o fornece uma carboxamida ou sulfonamida contendo compostos cã­clicos de fã³rmula (1), (1'), (100), (100'), (200) e (200') , , , , e e os enantiã´meros, diastereoisã´meros, tautã´meros, n-ã³xidos, solvatos e os sais farmaceuticamente aceitã¡veis dos mesmos.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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