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COMPOSE ACIDE DICARBOXYLIQUE
专利权人:
DAIICHI SANKYO COMPANY; LIMITED
发明人:
UTO, YOSHIKAZU,KATO, MIKIO,TAKAHASHI, HIDENORI,OGAWA, YASUYUKI,IWAMOTO,OSAMU,KONO, HIROKO,AOKI, KAZUMASA
申请号:
CA2909400
公开号:
CA2909400C
申请日:
2014.04.23
申请国别(地区):
CA
年份:
2017
代理人:
摘要:
It is an object of the present invention to provide amedicament for preventing or treating hyperphosphatemia.Solution: A compound having general formula (I) or apharmaceutically acceptable salt thereof.(see formula I)wherein:R1 is a C1-6 alkyl group, a C1-6 alkoxy C1-6 alkyl group, aC3-6 cycloalkyl group, or a C3-6 cycloalkyl C1-6 alkyl group;R2 is a hydrogen atom or a halogen group; R3 is a hydrogenatom, a halogen group, a halogeno C1-6 alkyl group, a halogenoC1-6 alkoxy group, a C2-5 saturated cyclic amino group, a C1-6dialkylamino group, a C3-6 cycloalkyl C1-6 alkoxy group or aC1-6 alkoxy group; A is a C3-6 cycloalkyl ring; X is CH or N;Y is CH or N; Z is CH or N; and n is 1, 2, 3 or 4.
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