Alexander Flohr;Jens-Uwe Peters;Konrad Bleicher;Rosa Maria Rodriguez-Sarmiento;Eric Vieira;Matthias Koerner;Bernd Kuhn;Katrin Groebke Zbinden
发明人:
Konrad Bleicher,Alexander Flohr,Katrin Groebke Zbinden,Matthias Koerner,Bernd Kuhn,Jens-Uwe Peters,Rosa Maria Rodriguez-Sarmiento,Eric Vieira
申请号:
US13005572
公开号:
US08470820B2
申请日:
2011.01.13
申请国别(地区):
US
年份:
2013
代理人:
摘要:
The invention is concerned with novel nitrogen-containing heteroaryl derivatives of formula (I)wherein R1, R2, R3, R4, R5, A1, A2, and Y are as defined in the description and in the claims, as well as physiologically acceptable salts and esters thereof. These compounds inhibit PDE10A and can be used as medicaments.