BAELL, JONATHAN BAYLDON,SLEEBS, BRAD,FLYNN, BERNARD LUKE,STREET, IAN PHILLIP,QUAZI, NURUL,BUI, CHINH THIEN
申请号：
ES07815371
公开号：
ES2399071T3
申请日:
2007.10.16
申请国别(地区):
ES
年份:
2013
代理人:
摘要：
A compound represented by formula (If) or a salt thereof: wherein X represents O or NR (where R is selected from H, alkyl, aryl, cycloalkyl, acyl, alkenyl, heterocyclyl, heteroaryl, oxisulfinilo , oxysulfonyl, sulfinyl, and sulfonyl) Y represents NR3R4 R represents H or alkyl each R is independently selected from H, carboxyl, cyano, dihalometoxi, halogen, hydroxy, nitro, pentahaloethyl, phosphono, phosphorylamino, phosphinyl, sulfo, trihaloetenilo, trihalometanotio, trihalomethyl, trihalomethoxy, acyl, acylamino, acylimino, aciliminoxi, acyloxy, arylalkyl , arylalkoxy, alkenyl, alkenyloxy, alkoxy, alkyl, alkynyl, alkynyloxy, amino, aminoacyl, aminoacyloxy, aminosulfonyl, aminotioacilo, aryl, arylamino, aryloxy, cycloalkenyl, cycloalkyl, heteroaryl, heterocyclyl, oxyacyl, oxyacylamino, oxiaciloxi, oxiacilimino, oxisulfinilamino, oxisulfonilamino , oxitioacilo, oxitioaciloxi, sulfinyl, sulfinylamino, sulfonyl, sulfonylamino, thio, thioacyl, and thioacylamino R1 represents cycloalkyl, cycloalkenyl, alkyl, acyl, aryl, heterocyclyl, or heteroaryl R2 represents H, cycloalkyl, alkyl, acyl, aryl, alkenyl, heterocyclyl, heteroaryl, oxisulfinilo, oxysulfonyl, sulfinyl, or sulfonyl R3 and R4 each independently represent alkyl, or together with the N atom N-containing heteroaryl or heterocyclyl containing N and wherein each acyl, acylamino, acylimino, aciliminoxi, acyloxy, arylalkyl, arylalkoxy, alkenyl, alkenyloxy, alkoxy, alkyl, alkynyl, alkynyloxy, amino, aminoacyl, aminoacyloxy, aminosulfonyl, aminotioacilo, aryl, arylamino, aryloxy, cycloalkenyl , cycloalkyl, heteroaryl, heterocyclyl, oxyacyl, oxyacylamino, oxiaciloxi, oxiacilimino, oxisulfinilamino, oxisulfonilamino, oxitioacilo, oxitioaciloxi, sulfinyl, sulfinylamino, sulfonyl, sulfonylamino, thio, thioacyl, and thioacylamino may be optionally substituted with one or more groups selected from hydroxyl, acyl, alkyl, alkoxy, alkenyl, alkenyloxy, alkynyl, alkynyloxy, amino, aminoacyl, thio, arylalkyl, arylalkoxy, aryl, ar
