OLIVIER GENESTE,JAMES BROOKE MURRAY,THIERRY LE DIGUARHER,ARNAUD LE TIRAN,JRME STARCK,ANNE BENOT - GUILLOUZIC,JAMES EDWARD PAUL FRANOISE - DAVIDSON,I CHEN,JEAN JEN - HENLIN,GUILLAUME MICHEL - DE NANTEU
申请号：
ARP140102712
公开号：
AR097008A1
申请日:
2014.07.22
申请国别(地区):
AR
年份:
2016
代理人:
摘要：
Claim 1: phosphate Compound of formula (1), in which X and y represent a carbon Atom or a nitrogen Atom, it being understood that no can simultaneously represent two carbon Atoms and two nitrogen Atoms； and a u00b9 a-squared form along with Atoms that are a Get an Aromatic heterocycle substituted het optionally or not, consisting of 5, 6 or 7 links.And they can contain, in addition to nitrogen or represented by X, and one to three heteroatoms selected irrespective of Oxygen, Sulfur and Nitrogen. The Nitrogen in question can be substituted with a group that represents a hydrogen Atom, an alkyl group C u2081 u208b u2086 linear or branched or a Group - C (o) - O - ALK in that ALK is a linear or branched alkyl group c u2081 u208b u2086,Or, a u00b9 a-squared and independently of one another represent a hydrogen Atom, a linear or branched polihal u00f3genoalquilo c u2081 u208b u2086, a linear or branched alkyl group c u2081 u208b u2086 or cycloalkyl； T represents a hydrogen Atom, a linear or branched alkyl c u2081 u208b u2086 REPL Optionally controlled with one to three Halogen ATOMS, an alkyl group c u2081 u208b u2084 - nr u00b9r u00b2,Alkyl group or a c u2081 u208b u2084 - or u2076； r u00b9 and independently of one another R u00b2 represent a hydrogen Atom or a c u2081 u208b u2086 linear or branched alkyl group, or r u00b9 and R u00b2 form with the nitrogen Atom to which they are United heterocicloalquilo r u00b3 represents an alkyl group； c u2081 u208b u2086 linear or branched, alquenilo c u2082 u208b u2086 linear or branched, alquinilo c u2082 u208b u2086 linear or branched, cycloalkyl,Cicloalquil c u2083 u208b u2081 u2080alquilo c u2081 u208b u2086 linear or branched, heterocicloalquilo, aryl or heteroaryl, provided that one or more carbon Atoms of the previous groups, or their optional substituents can be deuterated (n) (S)； r u2074 represents a heteroaryl, aryl Group, cicloal Chyle or linear or branched alkyl c u2081 u208b u2086, provided that one or more carbon A
