BLUMENFELD MARTA,COMPERE DELPHINE,AUTHIER JEAN MICHEL
申请号：
IN6249/CHENP/2008
公开号：
IN269394B
申请日:
2008.11.17
申请国别(地区):
IN
年份:
2015
代理人:
摘要：
PIPERIDINE DERIVATIVES AS HUMAN PAPILLOMA VIRUS INHIBITORS HPV inhibitors with formula (I) where Gl represents a hydrocarbonated bond or chain possibly substituted by one or two alkyl groups, G2 represents a group (see formula la+Ib) or R represents a hydrogen, an alkyl, halogenoalkyl, or a prodrug radical such as carbamate, acetyl or dialkylaminomelhyl, G represents a bond or a hydrocarbonated chain possibly substituted by one or two alkyls, W represents an oxygen or sulphur, Rl and R2 each represent a group chosen from among hydrogen, halogen, hydroxyl, thio, alkoxy, halogenoalkoxy, alkylthio, halogenoalkyithio, amino, monoalkylamino, dialkylamino, cycloalkyl, alkyl or halogenoalkyi, R3 represents an acid or a prodrug radical of the acid function or a bioisostere of the acid function, A represents an aryl, cycloalkyl, cycloalkenyl or a heterocycle, each possibly substituted, and B represents an aryl or a heterocycle with 6 chains, each possibly substituted, and pharmaceutically acceptable salts.
