SATHE, Dhananjay G.,DAS, Arijit,RAIKAR, Sanjay,SURVE, Yashwant S.,PANDIT, Bhushan S.
申请号:
EP17890544
公开号:
EP3565552A4
申请日:
2017.12.21
申请国别(地区):
EP
年份:
2020
代理人:
摘要:
The present invention relates to the novel key intermediate, 4-{4-[(5 S)-(Aminomethyl)-2-oxo-1,3-oxazolidin-3-yl]-phenyl}-morpholin-3-one perchlorate, in the synthesis of rivaroxaban. The invention further relates to the crystalline form of novel intermediate, the process to prepare the novel intermediate and method of preparing rivaroxaban using this novel intermediate. The invention provides an improved and efficient process for preparation of Rivaroxaban.