Kenneth W. Bair,Torsten Herbertz,Goss S. Kauffman,Katherine J. Kayser-Bricker,George P. Luke,Matthew W. Martin,David S. Millan,Shawn E. R. Schiller,Adam C. Talbot
申请号:
US14546775
公开号:
US09388161B2
申请日:
2014.11.18
申请国别(地区):
US
年份:
2016
代理人:
摘要:
The present invention relates to inhibitors of bromo and extra terminal (BET) bromodomains that are useful for the treatment of cancer, inflammatory diseases, diabetes, and obesity, having Formula I:wherein W, X, Y, Z, R1, R2, R5, and R8 are as described herein.