Bair, Kenneth W.,Herbertz, Torsten,Kauffman, Goss Stryker,Kayser-Bricker, Katherine J.,Luke, George P.,Martin, Matthew W.,Millan, David S.,Schiller, Shawn E.R.,Talbot, Adam C.
申请号：
EP14862604
公开号：
EP3071203A4
申请日:
2014.11.18
申请国别(地区):
EP
年份:
2017
代理人:
摘要：
The present invention relates to inhibitors of bromo and extra terminal (BET) bromodomains that are useful for the treatment of cancer, inflammatory diseases, diabetes, and obesity, having Formula I: wherein W, X, Y, Z, R1, R2, R5, and R8 are as described herein.
