Kenneth W. BAIR,Torsten HERBERTZ,Goss S. KAUFFMAN,Katherine J. KAYSER-BRICKER,George P. LUKE,Matthew W. MARTIN,David S. MILLAN,Shawn E.R. SCHILLER,Adam C. TALBOT
申请号:
US15153685
公开号:
US20160256448A1
申请日:
2016.05.12
申请国别(地区):
US
年份:
2016
代理人:
摘要:
The present invention relates to inhibitors of bromo and extra terminal (BET) bromodomains that are useful for the treatment of cancer, inflammatory diseases, diabetes, and obesity, having Formula I:wherein W, X, Y, Z, R1, R2, R5, and R8 are as described herein.