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Pharmaceutical composition comprising (1R, 4R) -6'-fluor-N, N-dimethyl-4-phenyl-4 ', 9'-dihydro-3'H-spiro [cyclohexane-1,1'-pyran [3, 4, b] indole] -4-amine and an anticonvulsant
专利权人:
Grünenthal GmbH
发明人:
FROSCH, Stefanie,LINZ, Klaus,CHRISTOPH, Thomas
申请号:
ES13723004
公开号:
ES2624220T3
申请日:
2013.05.16
申请国别(地区):
ES
年份:
2017
代理人:
摘要:
Pharmaceutical composition comprising: (a) a first pharmacologically active ingredient selected from the compound according to formula (I) and physiologically acceptable salts thereof ** Formula ** and (b) a second pharmacologically active ingredient that is a selected anticonvulsant between the group consisting of retigabine, lamotrigine, lacosamide, levetiracetam, carbamazepine, sultiamo, phenacemide, felbamate, topiramate, phenethuride, brivaracetam, selectracetam, zonisamide, stiripentol, beclamide, mexiletine, ralfinamide, methoxonabital, methylphenbital, meclothonabital, meclothonabital, meclothonabital, meclothonabital, meclothonabital, primalbital , phenytoin, valeric amino (diphenylhidantoin) acid, mefenitoin, phosphenytoin, parametadione, trimetadione, etadione, ethosuximide, fensuximide, mesuximide, clonazepam, lorazepam, diazepam, clobazam, oxcarbazepine, eslicarbazidapidamine, aminoprophyrinoxylamino, amino, progabide, thiagabine, and physiologically acceptable salts d and the sameComposición farmacéutica que comprende: (a) un primer ingrediente farmacológicamente activo seleccionado entre el compuesto de acuerdo con la fórmula (I) y sales fisiológicamente aceptables del mismo**Fórmula** y (b) un segundo ingrediente farmacológicamente activo que es un anticonvulsivo seleccionado entre el grupo consistente en retigabina, lamotrigina, lacosamida, levetiracetam, carbamazepina, sultiamo, fenacemida, felbamato, topiramato, feneturida, brivaracetam, selectracetam, zonisamida, estiripentol, beclamida, mexiletina, ralfinamida, metilfenobarbital, fenobarbital, primidona, barbexaclona, metarbital, etotoína, fenitoína, ácido amino(difenilhidantoin)valérico, mefenitoína, fosfenitoína, parametadiona, trimetadiona, etadiona, etosuximida, fensuximida, mesuximida, clonazepam, lorazepam, diazepam, clobazam, oxcarbazepina, eslicarbazepina, rufinamida, ácido valproico, valpromida, ácido γ- aminobutírico, progabida, tiagabina, y sales fisiológicamente aceptables de los mis
来源网站:
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