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NOVI KIRALNI N-ACIL-5,6,7,(8-SUBSTITUIRANI)-TETRAHIDRO-(1,2,4)TRIAZOLO (4,3-A)PIRAZINI KOT SELEKTIVNI NK-3 RECEPTOR ANTAGONISTI, FARMACEVTSKI SESTAVEK, IN POSTOPKI ZA UPORABO V NK-3 POSREDOVANIH MOTNJAH
专利权人:
Euroscreen S.A.
发明人:
HOVEYEDA Hamid,HOVEYEDA Hamid,DUTHEUIL Guillaume,DUTHEUIL Guillaume,FRASER Graeme,FRASER Graeme,ROY Marie-Odile,ROY Marie-Odile,EL BOUSMAQUI Mohamed,EL BOUSMAQUI Mohamed,BATT Frederic,BATT Frederic
申请号:
SI201230520
公开号:
SI2763992T1
申请日:
2012.10.03
申请国别(地区):
SI
年份:
2016
代理人:
摘要:
The present invention relates to novel compounds of Formula I and their use in therapeutic treatments. The invention further relates to a novel chiral synthesis of 5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines using N-sp3 protective groups. The invention also provides intermediates for use in the synthesis of compounds of Formula I.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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