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N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
专利权人:
Incyte Corporation;Incyte Holdings Corporation
发明人:
James D Rodgers,Stacey Shepard,Argyrios G Arvanitis,Haisheng Wang,Louis Storace,Beverly Folmer,Wenyu Zhu,Joseph Glenn,Lixin Shao
申请号:
US14250843
公开号:
US09334274B2
申请日:
2014.04.11
申请国别(地区):
US
年份:
2016
代理人:
摘要:
The present invention relates to N-(hetero)aryl-pyrrolidine derivatives of Formula I:which are JAK inhibitors, such as selective JAK1 inhibitors, useful in the treatment of JAK-associated diseases including, for example, inflammatory and autoimmune disorders, as well as cancer.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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