BARTOLOMÉ-NEBREDA,JOSÉ, MANUEL,CONDE-CEIDE,SUSANA,MACDONALD,GREGOR,JAMES,PASTOR-FERNÁNDEZ,JOAQUIN,VAN GOOL, MICHIEL, LUC, MARIA,MARTÍN-MARTÍN,MARÍA,LUZ,VANHOOF, GRETA, CONSTANTIA, PETER
申请号:
MYPI 2012003971
公开号:
MY160305A
申请日:
2011.03.08
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
THE PRESENT INVENTION RELATES TO NOVEL IMIDAZO[1,2-A]PYRAZINE DERIVATIVES WHICH ARC INHIBITORS OF THE PHOSPHODIESTERASE 10 ENZYME (PDE 10) AND WHICH ARE USEFUL FOR THE TREATMENT OR PREVENTION OF NEUROLOGICAL, PSYCHIATRIC AND METABOLIC DISORDERS IN WHICH THE PDE10 ENZYME IS INVOLVED. THE INVENTION IS ALSO DIRECTED TO PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH COMPOUNDS, TO PROCESSES TO PREPARE SUCH COMPOUNDS AND COMPOSITIONS, TO THE USE OF SUCH COMPOUNDS OR PHARMACEUTICAL COMPOSITIONS FOR THE PREVENTION OR TREATMENT OF NEUROLOGICAL, PSYCHIATRIC AND METABOLIC DISORDERS AND DISEASES.