GERLACH, MATTHIAS,SEIPELT, IRENE,BLUMENSTEIN, LARS,MUELLER, GILBERT,GÜNTHER, ECKHARD,SCHUSTER, TILMANN,TEIFEL, MICHAEL
申请号：
ES12713705
公开号：
ES2552515T3
申请日:
2012.04.04
申请国别(地区):
ES
年份:
2015
代理人:
摘要：
A compound according to the general formula (I) ** Formula ** in which the substituents R1, R2, X have the following meaning: X is O R1 (I) substituted aryl, wherein the aryl group may be substituted with one or more F, CI, Br, I, CF3, CN, NH2, NH-alkyl, NH-cycloalkyl, NH-heterocyclyl, NH-aryl, NH-heteroaryl, NH-alkyl-cycloalkyl, NH-alkyl-heterocyclyl, NH -alkyl-aryl, NH-alkyl-heteroaryl, NH-alkyl-NH2, NH-alkyl-OH, N (alkyl) 2, NHC (O) -alkyl, NHC (O) -cycloalkyl, NHC (O) -heterocyclyl, NHC (O) -aryl, NHC (O) -heteroaryl, NHC (O) -alkyl-aryl, NHC (O) -alkyl-heteroaryl, NHSO2-alkyl, NHSO2-cycloalkyl, NHSO2-heterocyclyl, NHSO2-aryl, NHSO2- heteroaryl, NHSO2-alkyl-aryl, NHSO2-alkyl-heteroaryl, NO2, SH, S-alkyl, S-aryl, S-heteroaryl, OH, OCF3, O-alkyl, O-cycloalkyl, O-heterocyclyl, O-aryl, O-heteroaryl, O-alkyl-cycloalkyl, O-alkyl-heterocyclyl, O-alkyl-aryl, O-alkyl-heteroaryl, O-alkyl-OH, O- (CH2) nO, O - (- CH2-CH2-O -) n-CH2-CH2-OH, OC ( O) -alkyl, OC (O) -cycloalkyl, OC (O) -heterocyclyl, OC (O) -aryl, OC (O) -heteroaryl, OC (O) -alkyl-aryl, OC (O) -alkyl-heteroaryl , OC (O) -NH-alkyl, OSO3H, OSO2-alkyl, OSO2-cycloalkyl, OSO2-heterocyclyl, OSO2-aryl, OSO2-heteroaryl, OSO2-alkyl-aryl, OSO2-alkyl-heteroaryl, OP (O) (OH ) 2, C (O) -alkyl, C (O) -aryl, C (O) -heteroaryl, O- CO2-alkyl, CO2H, CO2-alkyl, CO2-cycloalkyl, CO2-heterocyclyl, CO2-aryl, CO2- heteroaryl, CO2-alkyl-cycloalkyl, CO2-alkyl-heterocyclyl, CO2-alkyl-aryl, CO2-alkyl-heteroaryl, C (O) -NH2, C (O) NH-alkyl, C (O) NHcycloalkyl, C (O ) NH-heterocyclyl, C (O) NH-aryl, C (O) NH-heteroaryl, C (O) NH-alkylcycloalkyl, C (O) NH-alkylheterocyclyl, C (O) NH-alkyl-aryl, C (O) NH-alkyl-heteroaryl, C (O) N (alkyl) 2, C (O) N (cycloalkyl) 2, C (O) N (aryl) 2, C (O) N (heteroaryl) 2, SO -alkyl, SO-aryl, SO2-alkyl, SO2-heterocyclyl； SO2-aryl, SO2NH2, SO2NH-alkyl, SO2NH-aryl, SO2NH-heteroaryl, SO2NH-alkyl-aryl, SO3H, SO2O-alkyl, SO2O-aryl, SO2O-alkyl-aryl, alkyl, cycloalkyl, heterocyclyl, aryl or heteroaryl the same or dif
