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COMPOSES DE TYPE PYRAZOL-4-YL-HETEROCYCLYL-CARBOXAMIDE ET LEURS METHODES D'UTILISATION
专利权人:
F. HOFFMANN-LA ROCHE AG;F.HOFFMANN-LA ROCHE AG
发明人:
HODGES, ALASTAIR J.,MATTEUCCI, MIZIO,SHARPE, ANDREW,SUN, MINGHUA,TSUI, VICKIE H.,WANG, XIAOJING
申请号:
CA2845191
公开号:
CA2845191A1
申请日:
2012.09.26
申请国别(地区):
CA
年份:
2013
代理人:
摘要:
Pyrazol-4-yl-heterocyclyl-carboxamide compounds of Formula (I), including stereoisomers, geometric isomers, tautomers, and pharmaceutically acceptable salts thereof, wherein X is a thiazolyl, pyrazinyl, pyridinyl, or pyrimidinyl, are useful for inhibiting Pim kinase, and for treating disorders such as cancer mediated by Pim kinase. Methods of using compounds of Formula (I), for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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