КИСС Ласло Эрно (PT),ЛИРМОНТ Дэвид Александр (PT),РОЗА Карла Патрисиа да Кошта Перейра (PT),ГУЖМАН ДЕ НОРОНЬЯ Рита (PT),ПАЛЬМА Педро Нуно Леаль (PT),СУАРИШ ДА СИЛЬВА Патрисиу Мануэль Виейра Араужу (PT
申请号：
RU2011129416/04
公开号：
RU2011129416A
申请日:
2009.12.23
申请国别(地区):
RU
年份:
2013
代理人:
摘要：
1. The compound having formula I or formula II: where R1 and R2 can each be independently selected from H, C-alkyl, C-alkoxy, aryl, heteroaryl, partially or fully saturated heterocyclyl, C-cycloalkyl, aryl-C-alkyl , heteroaryl-C-alkyl, heterocyclyl-C-alkyl, C-cycloalkyl-C-alkyl, R1a, halogen, OH, OR1a, OCOR1a, SH, SR1a, SCOR1a, NH, NHR1a, NHSONH, NHSOR1a, NR1aCOR1b, NHCOR1a, , COR1a, CSR1a, CN, COOH, COOR1a, CONH, CONHOH, CONHR1a, CONHOR1a, SOR1a, SOH, SONH, CONR1aR1b, SONR1aR1b, where R1a and R1b are independently selected from C-alkyl, substituted C-alkylaryl, aryl, -cycloalkyl and heterocyclyl, or R1a and R1b, together with heteroatoms m to which they are attached can form heterocyclyl, where when R1 or R2 is C-alkyl, alkoxy, aryl, heteroaryl, heterocyclyl, C-cycloalkyl, aryl-C-alkyl, heteroaryl-C-alkyl, heterocyclyl-C -alkyl, C-cycloalkyl-C-alkyl, C-alkyl, C-cycloalkyl or represents a group containing one or more of these components, each of these components may be optionally substituted by one or more groups selected from R1c, halogen, aryl, heteroaryl, heterocyclyl, C-alkoxy, aryloxy, heteroaryloxy, heterocyclyloxy, and yl-C-alkyl, heteroaryl-C-alkyl, heterocyclyl-C-alkyl, C-cycloalkyl-C-alkyl, aryl-C-alkoxy, heteroaryl-C-alkoxy, heterocyclyl-C-alkoxy, C-alkylamine, C- dialkylamine, C-alkyl, OH, OR1c, OCOR1c, SH, SR1c, SCOR1c, NH, NO, NHR1c, NHSONH, NHSOR1c, NR1cCOR1d, NHC (NH) NH, NHCOR1c, NR1cR1d, COR1c, CSR1c, CN, COOH, CONH, CONHOH, CONHR1c, CONHOR1c, C (NOH) NH, CONR1cR1d, SOR1c, SOH, SONH, SONR1cR1d, where R1c and R1d are independently selected from C-alkyl, substituted C-alkyl, aryl, heteroaryl, C-cycloalkyl, hetero or R1c and R1d, together with the heteroatom to which they are attached, can form heterocyclyl, where when the substituent at R1 or R2 is1. Соединение, имеющее формулу I или формулу II:где R1 и R2 каждый может быть независимо выбран из Н, С-алкила, C-алкокси, арила, гетероарила, частично или полностью насыщенного гетероциклила, С-циклоалкила
