您的位置: 首页 > 农业专利 > 详情页

Alpha-substituted glycinamide derivative
专利权人:
Kissei Pharmaceutical Co.; Ltd.
发明人:
HIRASAWA, Hideaki,KAWAMURA, Naohiro,KOBAYASHI, Junichi
申请号:
ES14794817
公开号:
ES2645847T3
申请日:
2014.05.07
申请国别(地区):
ES
年份:
2017
代理人:
摘要:
A compound represented by the general formula (I) or a pharmaceutically acceptable salt thereof: ** Formula ** wherein: A1 is a group selected from the group consisting of the following a) to c): a) C6-C10 aryl, wherein the anyl is not substituted or is substituted with 1 to 2 substituents independently selected from the group consisting of the following: a halogen atom, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 haloalkyl, C1- haloalkoxy C6, (C1-C6) alkoxycarbonyl, cyano, C1-C6 hydroxyalkyl, carbamoyl, nitro, amino, (C1-C6) alkoxylamino-C1-C6 alkyl, mono (di) (C1-C6) alkyl, amino ( C1-C6) carbonylamino, (C1-C6) alkyl sulfonylamino and (C1-C6) sulfonyl, b) 5-membered heterocycle, wherein the anyl is not substituted or is substituted with 1 to 2 substituents independently selected from the group consisting in the following: a halogen, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 haloalkyl, cyano and C1-C6 haloalkoxy atom, and c) 6-membered heterocycle, wherein the anyl is unsubstituted or substituted with 1 to 2 substituents independently selected from the group consisting of the following: a halogen atom, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 haloalkyl, cyano and C1-C6 haloalkoxy; A2 is a group selected from the group consisting of the following d) af): d) C6-C10 aryl, wherein the anyl is not substituted or is substituted with 1 to 2 substituents independently selected from the group consisting of the following: a halogen atom, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 hydroxyalkoxy, C1-C6 haloalkyl, C1-C6 haloalkoxy, cyano, amino, nitro, carboxy, (C1-C6) carbonylamino, (C1-alkyl) -C6) carbonyloxy, (C1-C6) alkylcarbonyl and (C7-C10) oxycarbonyl, e) heterocycle, wherein the anyl is not substituted or is substituted with 1 to 2 substituents independently selected from the group consisting of the following: a halogen atom, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 haloalkyl, C1-C6 haloalkoxy, cyano, mono (di) alkyl (C1-C6) amino, (C1-C6) alkyl sulfanyl, amino , aralkyl
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充