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HETEROCYCLIC COMPOUNDS AS CCR2B ANTAGONISTS
专利权人:
ASTRAZENECA AB
发明人:
JUSTIN FAIRFIELD BOWER,JEFFREY PHILIP POYSER,PAUL TURNER,DAVID WATERSON,JON WINTER
申请号:
MYPI 20056171
公开号:
MY147400A
申请日:
2005.12.22
申请国别(地区):
MY
年份:
2012
代理人:
摘要:
296 ABSTRACT TITLE: ME'RHOD 5 COMPOUNDS OFFONNULA (1) Q- L -W- C(=X) - Z - P I 0 WHEREIN Q IS AN ARNINE OF THE FORMULA -N(R')(R 2). L IS AN ALKV] OR LICTEROCYCLYL-ALKVI LINKER; W IS A 6- OR 7-MEMBERED ALIPHATIC RING COMPRISING RING ATORNS Y' AND Y2 WHICH ARE LINKED TO GROUPS L AND C(X) RESPECTIVELV AND Y' AND Y2 ARE INDEPENCLENTLY SELECTED FROM N AND C; 1 5 X IS 0, N, N-CN OR S; Z IS NR 3 P IS AN OPTIONALLY SUBSTITUTED NIONOCYCLIC OR BICYCLIC ARYL OR HETEROARYL GROUP AND PHARMACEUTICALLY ACCEPTABLE SALTS OR SOLVATES THEREOF, ARE USEFUL IN THE TREATMENT OF C-C CHERNOKINE MEDIATED CONDITIONS. 20
来源网站:
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