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Fluoroindole derivatives as muscarinic M1 receptor positive allosteric modulators
专利权人:
Suven Life Sciences Limited
发明人:
NIROGI Ramakrishna,SHINDE Anil Karbhari,MOHAMMED Abdul Rasheed,SUBRAMANIAN Ramkumar,BENADE Vijay Sidram,BHYRAPUNENI Gopinadh,JASTI Venkateswarlu
申请号:
MDE20180689
公开号:
MD3347349T2
申请日:
2016.07.19
申请国别(地区):
MD
年份:
2019
代理人:
摘要:
This invention refers to compounds of formula (I) or their isotopic forms, stereoisomers or acceptable farmaceous salts, as positive modulators of muscle receptors M1 (M1 PAM). This invention also describes the pharmaceutical compositions containing these compounds and their use in the treatment of the various diseases selected from schizophrenia, cognitive disorders, duelling or sleep disorders, in the positive allosteric modulation of the muscarinic receptor M1.(Formula I)Prezenta invenţie se referă la compuşi din formula (I) sau formele lor izotopice, stereoizomerii sau sărurile acceptabile farma-ceutic, ca modulatori alosterici pozitivi ai receptorilor muscarinici M1 (M1 PAM). Prezenta invenţie descrie de asemenea compoziţii farmaceutice care conţin compuşii respectivi şi utilizarea acestora în tratamentul diferitelor afecţiuni selectate dintre schizofrenie, tulburări cognitive, duerere sau tulburări de somn, în modularea alosterică pozitivă a receptorului muscarinic M1.(Formula I)
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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