Disclosed are a novel rebamipide prodrug, a method for preparing thesame, and use thereof. Also, a pharmaceutical composition comprising thenovel rebamipide prodrug as an active ingredient is provided. therebamipide prodrug is increased 25-fold in absorption rate compared to rebamipide itself, and can be applied to theprophylaxis or therapy of gastric ulcer, acute gastritis, chronic gastritis, xerophthalmia, cancer, osteoarthritis, rheumatoid arthritis, or obesity.一種以新穎的瑞巴派特前體藥物作為活性成分之藥物組成，與瑞巴派特比較，此瑞巴派特前體藥物在吸收率上係增加25倍，且可以做為胃潰瘍、急性胃炎、慢性胃炎、乾眼症、癌症、骨關節炎、類風溼性關節炎、與肥胖的預防與治療。
