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FORMES CRISTALLINES DE TEBIPENEME PIVOXIL, COMPOSITIONS LES CONTENANT, PROCEDES DE FABRICATION ET D'UTILISATION
专利权人:
SPERO THERAPEUTICS; INC.
发明人:
JAIN, AKASH,HECKER, EVAN,EDWARDS, RICHARD,BONNAUD, THIERRY
申请号:
CA3049690
公开号:
CA3049690A1
申请日:
2018.02.06
申请国别(地区):
CA
年份:
2018
代理人:
摘要:
The disclosure is directed to new crystalline tebipenem pivoxil salt forms, including a crystalline tebipenem pivoxil ethane sulfonate salt form (Form A), a crystalline tebipenem pivoxil ketoglutarate salt form (Form A), tebipenem pivoxil maleate salt forms (Form A and Form B), a tebipenem pivoxil malate salt form (Form A), a tebipenem pivoxil methane sulfonate salt form (Form B), a tebipenem pivoxil hydrobromide salt form (Form B), and a tebipenem pivoxil edisylate salt form (Form A). The disclosure also includes a composition, comprising a crystalline tebipenem pivoxil salt and a pharmaceutically acceptable carrier and further includes a method for treating an antibiotic resistant bacterial infection, comprising administering to a patient in need of such treatment a therapeutically effective amount of a crystalline tebipenem pivoxil salt.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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