SILVANA MARCEL LEIT DE MORADEI,GERALDINE C. HARRIMAN,JEREMY ROBERT GREENWOOD,SHOMIR GHOSH
申请号：
ARP160103591
公开号：
AR106799A1
申请日:
2016.11.23
申请国别(地区):
AR
年份:
2018
代理人:
摘要：
Useful ester compounds as acetyl CoA carboxilasa (ACC) inhibitorsTheir composition and methods for plant protection and treatment of human infection. Page: 1 1. Claim 1: a formula compound (1),Or a medically acceptable salt or an agricultural acceptable salt, wherein:- yes.I am me!R¹ is hydrogen or aliphatic C₁₋₄ optionally substituted with 1-4 halogens independently selected from halogen, -OR, -SR, -N (R) ₂,-N (R) C (O) R -C (O) N (R)-N (R) C (O) N (R)-N (R) C (O) OR -OC (O) N (R)-N (R) S (O) R -S (O) N (R)-C (o) r, - C (o) o r, - OC (o) r, O-S (o) 8322； R 2 is r7491；R8310a each,R831181 and r831220 independent oxo, halogen, CN, r74919；-OR -SR -N (R)-N (R) C (O) R -C (O) N (R)-N (R) C (O) N (R)-N (R) C (O) OR -OC (O) N (R)-N (R) S (O) R -S (O) N (R)-C (O) R, -C (O) OR, -OC (O) R, -S (O) R, or -S (O) ₂R； each R is independently hydrogen, or Rᵃ；each Rᵃ is independently an optionally substituted group selected from aliphatic C₁₋₆,A saturated or partially unsaturated 3-8 member single cycle ring, a phenyl, an 8-10 member double cycle ring, a saturated or partially unsaturated single cycle ring, which is composed of 4-8 members and has 1-2 nitrogen and oxygen free heteroatoms, O sulfur, a 5-6 member single ring aromatic ring, consisting of 1-4 heteroatoms without nitrogen, oxygen or sulfur, or an 8-10 member double ring heteroaromatic ring, consisting of 1-5 heteroatoms independently selected from nitrogen, oxygen or sulfur； This is a covalent link,a. L2 is a covalent link or a bivalent or branched hydrogen carbon chain of 1-6 members, in which L2 is replaced by r8313；R es -OR -C (O) OR -N (R) C (O) OR -OC (O) N (R)-C (O) N (R) OR -C (O) NH-C (O) NHR-C (O) N (R)O-C (o) hy is a saturated or partially unsaturated single ring, which consists of 3-8 members and 1-2 heteroatoms selected independently from nitrogen, oxygen or sulfur. It is a 5-6 member single ring aromatic ring, which consists of 1-4 non nitrogen atoms, a. Oxygen or sulfur, or 8-10 member bicyclic heteroaromat
