您的位置: 首页 > 农业专利 > 详情页

hydroxy quinoline compound and pharmaceutical formulation
专利权人:
S.A.;Polichem
发明人:
Frederico Mailland,Michela Legora,Stefania Gagliardi
申请号:
BR112012015728
公开号:
BR112012015728A2
申请日:
2010.12.28
申请国别(地区):
BR
年份:
2019
代理人:
摘要:
hydroxy quinoline compound and pharmaceutical formulation. The present invention provides novel tertiary 8-hydroxy-quinoline-7-carboxamide derivatives of formula (I) and pharmaceutically acceptable salts thereof. These compounds are useful as antifungal agents. specifically, these compounds were tested against tricophyton rubrum, tricophyton mentagrophytes, aspergillus niger and bravicaulis scopulariopsis. These compounds are also active against candida species such as candida albicans and candida glabrata.composto de hidróxi-quinolina e formulação farmacêutica. a presente invenção fornce novos derivados terciários de 8-hidróxi-quinolina-7-carboxamida de fórmula geral (i) e sais farmaceuticamente aceitáveis destes. estes compostos são úteis como agentes antifúngicos. especificamente, estes compostos foram testados contra tricophyton rubrum, tricophyton mentagrophytes, aspergillus niger e bravicaulis scopulariopsis. esses compostos são também ativos contra espécies de candida, tais como candida albicans e candida glabrata.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充