4-(8-METHOXY-1-((1-METHOXYPROPAN-2-YL)-2-(TETRAHYDRO-2H-PYRAN-4-YL)-1 H-IMIDAZO[4,5-C]QUINOLIN-7-YL)-3,5-DIMETHYLISOXAZOLE ET UTILISATION DE CE DERNIER EN TANT QU'INHIBITEUR DE BROMODOMAINES
- 专利权人:
- GLAXOSMITHKLINE LLC
- 发明人:
- DEMONT, EMMANUEL HUBERT,JONES, KATHERINE LOUISE,WATSON, ROBERT J.
- 申请号:
- CA2843537
- 公开号:
- CA2843537A1
- 申请日:
- 2012.08.15
- 申请国别(地区):
- CA
- 年份:
- 2013
- 代理人:
- 摘要:
- Novel quinoline compounds of formula (I), pharmaceutical compositions containing such compounds and their use in therapy, as bromodomain inhibitors.
- 来源网站:
- 中国工程科技知识中心
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- 4-(8-METHOXY-1-((1-METHOXYPROPAN-2-YL)-2-(TETRAHYDRO-2H-PYRAN-4-YL)-1 H-IMIDAZO[4,5-C]QUINOLIN-7-YL)-3,5-DIMETHYLISOXAZOLE AND ITS USE AS BROMODOMAIN INHIBITOR
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