4-(8-METHOXY-1-((1-METHOXYPROPAN-2-YL)-2-(TETRAHYDRO-2H-PYRAN-4-YL)-1 H-IMIDAZO[4,5-C]QUINOLIN-7-YL)-3,5-DIMETHYLISOXAZOLE ET LEUR UTILISATION COMME INHIBITEUR DE BROMODOMAIN
- 专利权人:
- GlaxoSmithKline LLC
- 发明人:
- 申请号:
- EP16192662.1
- 公开号:
- EP3150601A1
- 申请日:
- 2012.08.15
- 申请国别(地区):
- EP
- 年份:
- 2017
- 代理人:
- 摘要:
- Novel quinoline compounds (I),pharmaceutical compositions containing such compounds and their use as bromodomain inhibitors in therapy.
- 来源网站:
- 中国工程科技知识中心
相关发明人
相关专利
- 4-(8-METHOXY-1-((1-METHOXYPROPAN-2-YL)-2-(TETRAHYDRO-2H-PYRAN-4-YL)-1 H-IMIDAZO[4,5-C]QUINOLIN-7-YL)-3,5-DIMETHYLISOXAZOLE AND ITS USE AS BROMODOMAIN INHIBITOR
- 4-(8-METHOXY-1-((1-METHOXYPROPAN-2-YL)-2-(TETRAHYDRO-2H-PYRAN-4-YL)-1 H-IMIDAZO[4,5-C]QUINOLIN-7-YL)-3,5-DIMETHYLISOXAZOLE ET UTILISATION DE CE DERNIER EN TANT QU'INHIBITEUR DE BROMODOMAINES
- 4 - (2 - 8 - metoxipropan - il) - 2 - (Tetrahydro - 2H - piran - 4-yl) - 1H imidazo [4,5-c] quinolin-1 - 7 - yl) - 3.5 - dimetilisoxazol as inhibitor of bromodomain and its use
- 4 - (4 - methoxy - (1 - (1 - metoxipropan - 2 - 2 - (IL) - tetrahydro - 2H - piran - 4-yl) - 1H imidazo [4,5-c] quinolin-1 - 7 - yl) - 3.5 - dimetilisoxazol as inhibitor of bromodomain and its use
- 4-(8-MÉTHOXY-1-((1-MÉTHOXYPROPAN-2-YL)-2-(TÉTRAHYDRO-2H-PYRAN-4-YL)-1 H-IMIDAZO[4,5-C]QUINOLIN-7-YL)-3,5-DIMÉTHYLISOXAZOLE ET UTILISATION DE CE DERNIER EN TANT QU'INHIBITEUR DE BROMODOMAINES