{2- [1- (3,5-Bis-trifluoromethyl-benzyl) -5-pyridin-4-yl-1H- [1,2,3] triazol-4-yl] -pyridin-3-yl} Novel intermediates and methods useful in the preparation of-(2-chlorophenyl) -methanone

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专利权人:

イーライ リリー アンド カンパニー

发明人:

マイケル・エドワード・コビアースキー,マイケル・イー・コパッチ,ピンユン・チェン

申请号：

JP2009543027

公开号：

JP5443168B2

申请日:

2007.12.04

申请国别(地区):

JP

年份:

2014

代理人:

摘要：

The present invention relates to novel compounds, (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone benzoate, and (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone toluate, which are useful intermediates for the preparation of the compound of Formula I: (I) The present invention further relates to novel processes for preparing a crystalline compound, which is {2-[1-(3,5-bis-trifluoromethyl-benzyl)-5-pyridin-4-yl-1H-[1,2,3]triazol-4-yl]-pyridin-3-yl}-(2-chlorophenyl)-methanone, Form IV.

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