Franco Bernini,Maria Pia Adorni,Pier Giorgio Petronini,Roberta Alfieri,Maricla Galetti,Elda Favari,Matteo Incerti
申请号：
US15501463
公开号：
US20170224647A1
申请日:
2015.08.03
申请国别(地区):
US
年份:
2017
代理人:
摘要：
New inhibitors of the activity of the multidrug resistance receptor 1 (MDR1), which are highly active to the MDR1 transporter, and showing a medium/high selectivity to such transporter, described by the structural formula (I): where R is a C1-C4 alkylene, optionally substituted with a C1-C3 alkyl. Said inhibitors are useful in the treatment or prevention of multi-drug resistance.
