您的位置: 首页 > 农业专利 > 详情页

AMINOPYRAZINE COMPOUNDS WITH A2A ANTAGONISTIC PROPERTIES
专利权人:
МЕРК ШАРП И ДОУМ КОРП. (US)
发明人:
КУАН Жунцзе (US),ТИНГ Полин (US),АЛИ Амджад (US),У Хэпин (US),БЕРЛИН Майкл (US),СТЭМФОРД Эндрю (US),ВАН Хунву (US),ЧЖОУ Ган (US),КИМ Дэвид (US),ДЭН Цяолинь (US),ЛИМ Йеон-Хее (US),ЮЙ Юнун (US)
申请号:
RU2017120853
公开号:
RU2017120853A
申请日:
2015.11.13
申请国别(地区):
RU
年份:
2018
代理人:
摘要:
Disclosed are compounds of Formula A and Formula A-1, or a salt thereof, and pharmaceutical formulations (pharmaceutical compositions) comprising those compounds, or a salt thereof; wherein "R1", "RA-1", "R2", "R3", and "Het" are defined herein above, which compounds are believed suitable for use in selectively antagonizing the A2a receptors, for example, those found in high density in the basal ganglia. Such compounds and pharmaceutical formulations are believed to be useful in treatment or management of neurodegenerative diseases, for example, Parkinson's disease, or movement disorders arising from use of certain medications used in the treatment or management of Parkinson's disease.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充