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COMPOSÉ DE PYRAZOLE
专利权人:
Dainippon Sumitomo Pharma Co.; Ltd.
发明人:
申请号:
EP11806858.4
公开号:
EP2594559A1
申请日:
2011.07.14
申请国别(地区):
EP
年份:
2013
代理人:
摘要:
The present invention relates to a novel serotonin reuptake inhibitor which also exhibits 5-HT2 C antagonistic action (antidepressive and anxiolytic effects), in particular, 5-HT2 C inverse agonistic action comprising Compound (1) :or a pharmaceutically acceptable salt thereofwherein R1, R2 , R3 and R4 are independently hydrogen or C1-6 alkyl etc.; R5 is C4-7 alkyl or -(CR8R9)r-E; R6, R7, R8 and R9 are independently hydrogen, fluorine or C1-6 alkyl; A is C6-10 aryl or heteroaryl etc.; r is 1, 2, 3 or 4; E is C3-8 cycloalkyl or C6-10 aryl etc.; L is oxygen, sulfur or -NR10 -; n is 1, 2 or 3; R10 is hydrogen or C1-6 alkyl etc.; and X is hydrogen or halogen etc.
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